• 3159 Citations
  • 31 h-Index
1979 …2019

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Article
2019

1,2-Dihydrochromeno[2,3-c]pyrrol-3-one Derivatives: Synthesis and HPLC-ECD Analysis

Tóth, L., Kiss-Szikszai, A., Vasvári, G., Fenyvesi, F., Vecsernyés, M., Mátyus, P., Antus, S., Mándi, A. & Kurtán, T., jan. 1 2019, In : Synlett. 30, 7, p. 799-803 5 p.

Research output: Article

3 Citations (Scopus)

Chemically modified derivatives of the activator compound cloxyquin exert inhibitory effect on TRESK (K2P18.1) background potassium channel

Lengyel, M., Erdélyi, F., Pergel, E., Bálint-Polonka, Á., Dobolyi, A., Bozsaki, P., Dux, M., Király, K., Hegedüs, T., Czirják, G., Mátyus, P. & Enyedi, P., jan. 1 2019, In : Molecular pharmacology. 95, 6, p. 652-660 9 p.

Research output: Article

1 Citation (Scopus)
2018
8 Citations (Scopus)

HPLC-ECD and TDDFT-ECD study of hexahydropyrrolo[1,2-a]quinoline derivatives

Tóth, L., Mándi, A., Váradi, D., Kovács, T., Szabados, A., Kiss-Szikszai, A., Gong, Q., Zhang, H., Mátyus, P., Antus, S. & Kurtán, T., júl. 2018, In : Chirality. 30, 7, p. 866-874 9 p.

Research output: Article

5 Citations (Scopus)
2017

Remarkable regioselectivities in the course of the synthesis of two new Luotonin A derivatives

Atia, M., Bogdán, D., Brügger, M., Haider, N. & Mátyus, P., jan. 1 2017, In : Tetrahedron. 73, 23, p. 3231-3239 9 p.

Research output: Article

12 Citations (Scopus)

Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B

Meleddu, R., Distinto, S., Cirilli, R., Alcaro, S., Yanez, M., Sanna, M. L., Corona, A., Melis, C., Bianco, G., Mátyus, P., Cottiglia, F. & Maccioni, E., dec. 1 2017, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 32, 1, p. 264-270 7 p.

Research output: Article

9 Citations (Scopus)
2016

A novel 3-(4,5-diphenyl-1,3-oxazol-2-yl)propanal oxime compound is a potent Transient Receptor Potential Ankyrin 1 and Vanilloid 1 (TRPA1 and V1) receptor antagonist

Payrits, M., Sághy, Mátyus, P., Czompa, A., Ludmerczki, R., Deme, R., Sándor, Z., Helyes, Z. & Szoke, jún. 2 2016, In : Neuroscience. 324, p. 151-162 12 p.

Research output: Article

12 Citations (Scopus)

Dietary Phenolic Compounds Interfere with the Fate of Hydrogen Peroxide in Human Adipose Tissue but Do Not Directly Inhibit Primary Amine Oxidase Activity

Carpéné, C., Hasnaoui, M., Balogh, B., Matyus, P., Fernández-Quintela, A., Rodríguez, V., Mercader, J. & Portillo, M. P., jan. 1 2016, In : Oxidative medicine and cellular longevity. 2016, 2427618.

Research output: Article

9 Citations (Scopus)

Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida

Meleddu, R., Distinto, S., Corona, A., Maccioni, E., Arridu, A., Melis, C., Bianco, G., Mátyus, P., Cottiglia, F., Sanna, A. & De Logu, A., jan. 7 2016, (Accepted/In press) In : Journal of Enzyme Inhibition and Medicinal Chemistry. p. 1-6 6 p.

Research output: Article

5 Citations (Scopus)

Light-Enhanced Fluorescence of Multi-Level Cavitands Possessing Pyridazine Upper rim

Janosi, T. Z., Makkai, G., Kegl, T., Mátyus, P., Kollár, L. & Erostyak, J., márc. 1 2016, In : Journal of Fluorescence. 26, 2, p. 679-688 10 p.

Research output: Article

1 Citation (Scopus)
4 Citations (Scopus)

Novel (Hetero)arylalkenyl propargylamine compounds are protective in toxin-induced models of Parkinson's disease

Baranyi, M., Porceddu, P. F., Gölöncsér, F., Kulcsár, S., Otrokocsi, L., Kittel, A., Pinna, A., Frau, L., Huleatt, P. B., Khoo, M. L., Chai, C. L. L., Dunkel, P., Mátyus, P., Morelli, M. & Sperlágh, B., jan. 13 2016, (Accepted/In press) In : Molecular Neurodegeneration.

Research output: Article

19 Citations (Scopus)

One size does not fit all: Challenging some dogmas and taboos in drug discovery

Chai, C. L. L. & Mátyus, P., jan. 1 2016, In : Future Medicinal Chemistry. 8, 1, p. 29-38 10 p.

Research output: Article

6 Citations (Scopus)
6 Citations (Scopus)

Versatile synthesis of novel tetrahydroquinolines as potentially active semicarbazide-sensitive amine oxidase (SSAO) inhibitors via tert-Amino effect

Deme, R., Schlich, M., Mucsi, Z., Karvaly, G., Tóth, G. & Mátyus, P., szept. 21 2016, In : Arkivoc. 2016, 5, p. 164-196 33 p.

Research output: Article

3 Citations (Scopus)
2015

(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase

Meleddu, R., Distinto, S., Corona, A., Bianco, G., Cannas, V., Esposito, F., Artese, A., Alcaro, S., Matyus, P., Bogdan, D., Cottiglia, F., Tramontano, E. & Maccioni, E., márc. 26 2015, In : European Journal of Medicinal Chemistry. 93, p. 452-460 9 p.

Research output: Article

31 Citations (Scopus)

Analysis of Edg-Like LPA receptor-ligand interactions

Balogh, B., Pazmany, T. & Matyus, P., aug. 1 2015, In : Current pharmaceutical design. 21, 24, p. 3533-3547 15 p.

Research output: Article

Anti-inflammatory effects of a triple-bond resveratrol analog: Structure and function relationship

Antus, C., Radnai, B., Dombovari, P., Fonai, F., Avar, P., Matyus, P., Racz, B., Sumegi, B. & Veres, B., febr. 5 2015, In : European Journal of Pharmacology. 748, p. 61-67 7 p.

Research output: Article

18 Citations (Scopus)

Novel arylalkenylpropargylamines as neuroprotective, potent, and selective monoamine oxidase B inhibitors for the treatment of Parkinson's disease

Huleatt, P. B., Khoo, M. L., Chua, Y. Y., Tan, T. W., Liew, R. S., Balogh, B., Deme, R., Gölöncsér, F., Magyar, K., Sheela, D. P., Ho, H. K., Sperlágh, B., Mátyus, P. & Chai, C. L. L., febr. 12 2015, In : Journal of Medicinal Chemistry. 58, 3, p. 1400-1419 20 p.

Research output: Article

22 Citations (Scopus)
5 Citations (Scopus)

Water-soluble isoindolo[2,1-a]quinoxalin-6-imines: In vitro antiproliferative activity and molecular mechanism(s) of action

Parrino, B., Carbone, A., Ciancimino, C., Spanò, V., Montalbano, A., Barraja, P., Cirrincione, G., Diana, P., Sissi, C., Palumbo, M., Pinato, O., Pennati, M., Beretta, G., Folini, M., Matyus, P., Balogh, B. & Zaffaroni, N., ápr. 13 2015, In : European Journal of Medicinal Chemistry. 94, p. 149-162 14 p.

Research output: Article

36 Citations (Scopus)
2014

'Interrupted' diazotization of 3-aminoindoles and 3-aminopyrroles

Parrino, B., Spanò, V., Carbone, A., Montalbano, A., Barraja, P., Màtyus, P., Cirrincione, G. & Diana, P., jan. 1 2014, In : Tetrahedron. 70, 40, p. 7318-7321 4 p.

Research output: Article

7 Citations (Scopus)

Preparation of neuroprotective condensed 1,4-benzoxazepines by regio- And diastereoselective domino knoevenagel-[1,5]-hydride shift cyclization reaction

Tóth, L., Fu, Y., Zhang, H. Y., Mándi, A., Kövér, K. E., Illyés, T. Z., Kiss-Szikszai, A., Balogh, B., Kurtán, T., Antus, S. & Mátyus, P., nov. 6 2014, In : Beilstein Journal of Organic Chemistry. 10, p. 2594-2602 9 p.

Research output: Article

11 Citations (Scopus)
2013

CYP24A1 inhibition facilitates the anti-tumor effect of vitamin D3 on colorectal cancer cells

Kósa, J. P., Horváth, P., Wölfing, J., Kovács, D., Balla, B., Mátyus, P., Horváth, E., Speer, G., Takács, I., Nagy, Z., Horváth, H. & Lakatos, P., máj. 7 2013, In : World journal of gastroenterology. 19, 17, p. 2621-2628 8 p.

Research output: Article

22 Citations (Scopus)

Drug repositioning for treatment of movement disorders: From serendipity to rational discovery strategies

Bolgár, B., Arany, Á., Temesi, G., Balogh, B., Antal, P. & Mátyus, P., nov. 25 2013, In : Current topics in medicinal chemistry. 13, 18, p. 2337-2363 27 p.

Research output: Article

17 Citations (Scopus)

Imidazoline versus alpha2-adrenoceptors in the control of gastric motility in mice

Zádori, Z. S., Fehér, Á., Al-Khrasani, M., Lackó, E., Tóth, V. E., Brancati, S. B., Hein, L., Mátyus, P. & Gyires, K., ápr. 5 2013, In : European Journal of Pharmacology. 705, 1-3, p. 61-67 7 p.

Research output: Article

8 Citations (Scopus)

Lack of association between VAP-1/SSAO activity and corneal neovascularization in a rabbit model

Énzsöly, A., Markó, K., Tábi, T., Szöko, É., Zelkó, R., Tóth, M., Mark Petrash, J., Mátyus, P. & Németh, J., jún. 1 2013, In : Journal of neural transmission. 120, 6, p. 969-975 7 p.

Research output: Article

5 Citations (Scopus)

Multi-aspect candidates for repositioning: Data fusion methods using heterogeneous information sources

Arany, Á., Bolgár, B., Balogh, B., Antal, P. & Mátyus, P., jan. 1 2013, In : Current medicinal chemistry. 20, 1, p. 95-107 13 p.

Research output: Article

13 Citations (Scopus)
11 Citations (Scopus)

Temporal alteration of spreading depression by the glycine transporter type-1 inhibitors NFPS and Org-24461 in chicken retina

Kertesz, S., Szabo, G., Udvari, S., Levay, G., Matyus, P. & Harsing, L. G., jan. 25 2013, In : Brain research. 1492, p. 1-6 6 p.

Research output: Article

1 Citation (Scopus)
13 Citations (Scopus)
2012

Functionalization of the pyridazin-3(2H)-one ring via palladium-catalysed aminocarbonylation

Takács, A., Czompa, A., Krajsovszky, G., Mátyus, P. & Kollár, L., szept. 23 2012, In : Tetrahedron. 68, 38, p. 7855-7860 6 p.

Research output: Article

3 Citations (Scopus)
6 Citations (Scopus)

Novel 1,4-benzoxazine and 1,4-benzodioxine inhibitors of angiogenesis

Ilić, M., Ilaš, J., Dunkel, P., Mátyus, P., Boháč, A., Liekens, S. & Kikelj, D., dec. 1 2012, In : European Journal of Medicinal Chemistry. 58, p. 160-170 11 p.

Research output: Article

8 Citations (Scopus)

Study on the scope of tert-amino effect: New extensions of type 2 reactions to bridged biaryls

Bottino, P., Dunkel, P., Schlich, M., Galavotti, L., Deme, R., Regdon, G., Bényei, A., Pintye-Hódi, K., Ronsisvalle, G. & Mátyus, P., nov. 1 2012, In : Journal of Physical Organic Chemistry. 25, 11, p. 1033-1041 9 p.

Research output: Article

3 Citations (Scopus)
2011

3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A new scaffold for the selective inhibition of monoamine oxidase B

MacCioni, E., Alcaro, S., Cirilli, R., Vigo, S., Cardia, M. C., Sanna, M. L., Meleddu, R., Yanez, M., Costa, G., Casu, L., Matyus, P. & Distinto, S., szept. 22 2011, In : Journal of Medicinal Chemistry. 54, 18, p. 6394-6398 5 p.

Research output: Article

39 Citations (Scopus)

Lipase-catalyzed synthesis of both enantiomers of 3-chloro-1-arylpropan-1- ols

Pop, L. A., Czompa, A., Paizs, C., Toa, M. I., Vass, E., Mátyus, P. & Irimie, F. D., aug. 4 2011, In : Synthesis. 18, p. 2921-2928 8 p., T49711SS.

Research output: Article

3 Citations (Scopus)

Preliminary studies of the effects of vascular adhesion protein-1 inhibitors on experimental corneal neovascularization

Énzsöly, A., Dunkel, P., Récsán, Z., Gyorffy, H., Tóth, J., Marics, G., Bori, Z., Tóh, M., Zelkó, R., Di Paolo, M. L., Mátyus, P. & Németh, J., júl. 1 2011, In : Journal of neural transmission. 118, 7, p. 1065-1069 5 p.

Research output: Article

8 Citations (Scopus)

Suzuki-aza-Wittig, Suzuki-condensation and aza-Wittig-electrocyclic ring-closure tandem reactions for synthesis of fused nitrogen-containing ring systems

Krajsovszky, G., Károlyházy, L., Dunkel, P., Boros, S., Grillo, A. & Mátyus, P., szept. 21 2011, In : Arkivoc. 2011, 10, p. 229-253 25 p.

Research output: Article

Open Access
3 Citations (Scopus)

Synthesis and antiproliferative activity of 2-(([1,2,4]triazolo[4,3-b]- pyridazin-6-yloxy)methyl)-2,4-dimethyl-3,4-dihydro-2Hbenzo[b][1,4]oxazine derivatives

Ilić, M., Ilaš, J., Liekens, S., Mátyus, P. & Kikelj, D., okt. 23 2011, In : Arkivoc. 2011, 10, p. 298-311 14 p.

Research output: Article

4 Citations (Scopus)
7 Citations (Scopus)
2010

Alterations in brain extracellular dopamine and glycine levels following combined administration of the glycine transporter type-1 inhibitor Org-24461 and risperidone

Nagy, K., Marko, B., Zsilla, G., Matyus, P., Pallagi, K., Szabo, G., Juranyi, Z., Barkoczy, J., Levay, G. & Harsing, L. G., dec. 1 2010, In : Neurochemical research. 35, 12, p. 2096-2106 11 p.

Research output: Article

22 Citations (Scopus)

Cyclisation reactions of some pyridazinylimidoylketenes

Gaywood, A. P., Hill, L., Imam, S. H., McNab, H., Neumajer, G., O'Neill, W. J. & Mátyus, P., 2010, In : New Journal of Chemistry. 34, 2, p. 236-242 7 p.

Research output: Article

6 Citations (Scopus)

Reaction of chloropyridazin-3(2H)-ones with iodide ion. Part II

Károlyházy, L., Krajsovszky, G., Farkas, L., Boros, S., Csámpai, A. & Mátyusa, P., nov. 29 2010, In : Arkivoc. 2011, 2, 36991.

Research output: Article

1 Citation (Scopus)

SSAO substrates exhibiting insulin-like effects in adipocytes as a promising treatment option for metabolic disorders

Mercader, J., Iffiú-Soltesz, Z., Brenachot, X., Földi, Á., Dunkel, P., Balogh, B., Attané, C., Valet, P., Mátyus, P. & Carpéné, C., dec. 1 2010, In : Future Medicinal Chemistry. 2, 12, p. 1735-1749 15 p.

Research output: Article

16 Citations (Scopus)

Synthesis of novel fused azecine ring systems through application of the tert-amino effect

Dunkel, P., Túrós, G., Bényei, A., Ludányi, K. & Mátyus, P., márc. 27 2010, In : Tetrahedron. 66, 13, p. 2331-2339 9 p.

Research output: Article

39 Citations (Scopus)
4 Citations (Scopus)
24 Citations (Scopus)
2009

C-29 ecdysteroids from Ajuga reptans var. reptans

Ványolós, A., Simon, A., Tóth, G., Polgár, L., Kele, Z., Ilku, A., Mátyus, P. & Báthori, M., máj. 22 2009, In : Journal of Natural Products. 72, 5, p. 929-932 4 p.

Research output: Article

17 Citations (Scopus)