• 1813 Citations
  • 26 h-Index
20002019
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Research Output 2000 2019

  • 1813 Citations
  • 26 h-Index
  • 97 Article
  • 6 Review article
  • 1 Chapter
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Article
2019
Nitriles
Cycloaddition
Alkenes
Oxides
Cycloparaffins
1 Citation (Scopus)
Oxazoles
Heptanes
Capillary electrophoresis
Cyclodextrins
Capillary Electrophoresis
4 Citations (Scopus)
Open Access
Cell-Penetrating Peptides
Tight Junctions
Permeability
Cell Membrane
Claudin-4
2018
2 Citations (Scopus)

A De Novo Synthetic Route to 1,2,3,4-Tetrahydroisoquinoline Derivatives

Ábrahámi, R. A., Fustero, S., Fülöp, F. & Kiss, L., márc. 22 2018, (Accepted/In press) In : Synlett.

Research output: Article

Amination
Derivatives
1,2,3,4-tetrahydroisoquinoline
indene
4 Citations (Scopus)
Cyclohexenes
Cyclopentanes
Fluorination
Fluorine
Scaffolds
4 Citations (Scopus)

Niosomes decorated with dual ligands targeting brain endothelial transporters increase cargo penetration across the blood-brain barrier

Mészáros, M., Porkoláb, G., Kiss, L., Pilbat, A. M., Kóta, Z., Kupihár, Z., Kéri, A., Galbács, G., Siklós, L., Tóth, A., Fülöp, L., Csete, M., Sipos, Á., Hülper, P., Sipos, P., Páli, T., Rákhely, G., Szabó-Révész, P., Deli, M. A. & Veszelka, S., okt. 15 2018, In : European Journal of Pharmaceutical Sciences. 123, p. 228-240 13 p.

Research output: Article

Blood-Brain Barrier
Liposomes
Ligands
Brain
Endothelial Cells
2 Citations (Scopus)
Lactams
Ruthenium
Lactones
Scaffolds
Conservation
10 Citations (Scopus)

Selective Synthesis of Fluorine-Containing Cyclic β-Amino Acid Scaffolds

Kiss, L. & Fülöp, F., márc. 1 2018, In : Chemical Record. 18, 3, p. 266-281 16 p.

Research output: Article

Cyclic Amino Acids
Fluorine
Scaffolds
Amino acids
Derivatives
1 Citation (Scopus)

Stereocontrolled Synthesis of Fluorine-Containing Piperidine γ-Amino Acid Derivatives

Ouchakour, L., Ábrahámi, R. A., Forró, E., Haukka, M., Fülöp, F. & Kiss, L., jan. 1 2018, (Accepted/In press) In : European Journal of Organic Chemistry.

Research output: Article

Lactams
piperidine
Fluorine
fluorine
amino acids
2017
2 Citations (Scopus)

An Insight into Substrate-Dependent Fluorination of some Highly Substituted Alicyclic Scaffolds

Kiss, L., Petrovszki, Á., Vass, C., Nonn, M., Sillanpää, R., Haukka, M., Fustero, S. & Fülöp, F., jan. 1 2017, In : ChemistrySelect. 2, 10, p. 3049-3052 4 p.

Research output: Article

Fluorination
Scaffolds
Derivatives
Substrates
Cyclopentanes
3 Citations (Scopus)

Biotin and glutathione targeting of solid nanoparticles to cross human brain endothelial cells

Veszelka, S., Mészáros, M., Kiss, L., Kóta, Z., Páli, T., Hoyk, Z., Bozsó, Z., Fülöp, L., Tóth, A., Rákhely, G. & Deli, M. A., aug. 1 2017, In : Current Pharmaceutical Design. 23, 28, p. 4198-4205 8 p.

Research output: Article

Biotin
Nanoparticles
Glutathione
Endothelial Cells
Brain
5 Citations (Scopus)
Cyclic Amino Acids
Lactams
Enantiomers
enantiomers
amino acids
4 Citations (Scopus)

Fluorination of some highly functionalized cycloalkanes: Chemoselectivity and substrate dependence

Remete, A. M., Nonn, M., Fustero, S., Haukka, M., Fülöp, F. & Kiss, L., nov. 6 2017, In : Beilstein Journal of Organic Chemistry. 13, p. 2364-2371 8 p.

Research output: Article

Cycloparaffins
Fluorination
Cyclic Amino Acids
Stereoisomerism
Fluorine
7 Citations (Scopus)
Cycloparaffins
Fluorine
Scaffolds
Amines
Amino acids
7 Citations (Scopus)
Bearings (structural)
Furans
Cyclopentanes
Lactams
Ruthenium
2016
2 Citations (Scopus)

Anion-/cation-directed reaction routes to polymorphic forms of a pyrazole-type ligand and its coordination compounds with zinc. Key structural differences between polymorphs’

Barta Holló, B., Mészáros Szécsényi, K., Deli, M., Kiss, L., Kállay-Menyhárd, A., Živković-Radovanović, V. & Tomić, Z. D., jan. 7 2016, (Accepted/In press) In : Structural Chemistry. p. 1-13 13 p.

Research output: Article

Polymorphism
Anions
Cations
Zinc
zinc
6 Citations (Scopus)

A stereocontrolled protocol to highly functionalized fluorinated scaffolds through a fluoride opening of oxiranes

Remete, A. M., Nonn, M., Fustero, S., Fülöp, F. & Kiss, L., nov. 1 2016, In : Molecules. 21, 11, 1493.

Research output: Article

Epoxy Compounds
Fluorides
Scaffolds
fluorides
Cyclic Amino Acids
8 Citations (Scopus)

Chemoselective, Substrate-directed Fluorination of Functionalized Cyclopentane β-Amino Acids

Kiss, L., Nonn, M., Sillanpää, R., Haukka, M., Fustero, S. & Fülöp, F., dec. 6 2016, In : Chemistry - An Asian Journal. 11, 23, p. 3376-3381 6 p.

Research output: Article

Cyclopentanes
Fluorination
Halogenation
Amino Acids
Substrates
8 Citations (Scopus)

Cytotoxicity of different excipients on RPMI 2650 human nasal epithelial cells

Horváth, T., Bartos, C., Bocsik, A., Kiss, L., Veszelka, S., Deli, M., Újhelyi, G., Szabó-Révész, P. & Ambrus, R., máj. 1 2016, In : Molecules. 21, 5, 658.

Research output: Article

Excipients
Cytotoxicity
Nose
Cyclodextrins
Epithelial Cells
2 Citations (Scopus)
Cyclic Amino Acids
Carbamates
Polysaccharides
Derivatives
Amino Acids
2 Citations (Scopus)

Modulation of vascular reactivity by novel synthetic benzopyran analogues in rat aortas

Petrus, A., Sturza, A., Utu, D., Duicu, O., Bedreag, O., Kiss, L., Baczkó, I., Muntean, D. & Jost, N., 2016, In : Revista de Chimie. 67, 5, p. 908-910 3 p.

Research output: Article

Benzopyrans
Rats
Modulation
Muscle
Reactive Oxygen Species
33 Citations (Scopus)

Restraint stress-induced morphological changes at the blood-brain barrier in adult rats

Sántha, P., Veszelka, S., Hoyk, Z., Mészáros, M., Walter, F. R., Tóth, A. E., Kiss, L., Kincses, A., Oláh, Z., Seprényi, G., Rákhely, G., Dér, A., Pákáski, M., Kálmán, J., Kittel, A. & Deli, M., jan. 14 2016, In : Frontiers in Molecular Neuroscience. 8, JAN2016, 88.

Research output: Article

Blood-Brain Barrier
Claudin-5
Brain
Facilitative Glucose Transport Proteins
Frontal Lobe
5 Citations (Scopus)

Substrate-dependent fluorinations of highly functionalized cycloalkanes

Kiss, L., Remete, A. M., Nonn, M., Fustero, S., Sillanpää, R. & Fülöp, F., febr. 11 2016, In : Tetrahedron. 72, 6, p. 781-787 7 p.

Research output: Article

Cycloparaffins
Fluorination
Halogenation
Substrates
Lactams
11 Citations (Scopus)

Synthesis of fluorinated piperidine and azepane β-amino acid derivatives

Ábrahámi, R. A., Kiss, L., Barrio, P. & Fülöp, F., nov. 24 2016, In : Tetrahedron. 72, 47, p. 7526-7535 10 p.

Research output: Article

Derivatives
Amination
Amino Acids
Lactams
Stereoisomerism
2015
Cycloparaffins
Stereochemistry
Palladium
Iodides
Isomers
34 Citations (Scopus)

A novel and selective fluoride opening of aziridines by XtalFluor-E. synthesis of fluorinated diamino acid derivatives

Nonn, M., Kiss, L., Haukka, M., Fustero, S. & Fülöp, F., márc. 6 2015, In : Organic Letters. 17, 5, p. 1074-1077 4 p.

Research output: Article

Aziridines
Fluorides
fluorides
Derivatives
acids
4 Citations (Scopus)

Atp-sensitive potassium channel modulators and cardiac arrhythmias: An update

Muntean, D. M., Kiss, L., Jost, N. & Baczkó, I., jan. 1 2015, In : Current Pharmaceutical Design. 21, 8, p. 1091-1102 12 p.

Research output: Article

Potassium Channels
Cardiac Arrhythmias
Ischemia
KATP Channels
Physiological Stress
3 Citations (Scopus)
Atrial Fibrillation
Cardiac Arrhythmias
Heart Failure
Pharmacology
Therapeutics
4 Citations (Scopus)

Modulation of mitochondrial respiratory function and ROS production by novel benzopyran analogues

Petruş, A., Duicu, O. M., Sturza, A., Noveanu, L., Kiss, L., Dănilă, M., Baczkó, I., Muntean, D. M. & Jost, N., ápr. 15 2015, In : Canadian Journal of Physiology and Pharmacology. 93, 9, p. 811-818 8 p.

Research output: Article

Benzopyrans
Heart Mitochondria
Oxidative Phosphorylation
Reactive Oxygen Species
KATP Channels
8 Citations (Scopus)
Amino Acids
Lactams
Alkaloids
tashiromine
2-azetidinone
7 Citations (Scopus)

Preparation and investigation of mefenamic acid - polyethylene glycol - sucrose ester solid dispersions

Fülöp, I., Gyéresi, Á., Kiss, L., Deli, M., Croitoru, M. D., Szabó-Révész, P. & Aigner, Z., dec. 1 2015, In : Acta Pharmaceutica. 65, 4, p. 453-462 10 p.

Research output: Article

Mefenamic Acid
Sucrose
Esters
Solubility
Non-Steroidal Anti-Inflammatory Agents
22 Citations (Scopus)

Recent advances in the stereoselective syntheses of acyclic disubstituted β2,3-amino acids

Kiss, L., Cherepanova, M. & Fülöp, F., ápr. 8 2015, In : Tetrahedron. 71, 14, p. 2049-2069 21 p.

Research output: Article

Enantiomers
Amino Acids
5 Citations (Scopus)

Stereo- and regiocontrolled syntheses of exomethylenic cyclohexane β-amino acid derivatives

Kiss, L., Forró, E., Orsy, G., Ábrahámi, R. & Fülöp, F., nov. 27 2015, In : Molecules. 20, 12, p. 21094-21101 8 p.

Research output: Article

Lactams
cyclohexane
amino acids
Phosphoranes
analogs
17 Citations (Scopus)
metathesis
amino acids
Derivatives
Amino Acids
Stereochemistry
10 Citations (Scopus)
Lactams
Derivatives
Amino Acids
Cycloaddition
2-azetidinone
28 Citations (Scopus)

Supermacroporous chemically cross-linked poly(aspartic acid) hydrogels

Gyarmati, B., Mészár, E. Z., Kiss, L., Deli, M., László, K. & Szilágyi, A., aug. 1 2015, In : Acta Biomaterialia. 22, p. 32-38 7 p.

Research output: Article

Hydrogels
Aspartic Acid
Freezing
Acids
Gels
1 Citation (Scopus)

Ternary solid dispersions of oxicams: Dissolution and permeability study

Fülöp, I., Gyéresi, Á., Deli, M., Kiss, L., Croitoru, M. D., Szabó-Révész, P. & Aigner, Z., 2015, In : Farmacia. 63, 2, p. 286-295 10 p.

Research output: Article

tenoxicam
meloxicam
Permeability
Esters
Piroxicam
2014
14 Citations (Scopus)
Lactams
Enantiomers
enantiomers
amino acids
Derivatives
15 Citations (Scopus)

A selective synthesis of fluorinated cispentacin derivatives

Kiss, L., Nonn, M., Forró, E., Sillanpää, R., Fustero, S. & Fülöp, F., 2014, In : European Journal of Organic Chemistry. 2014, 19, p. 4070-4076 7 p.

Research output: Article

Lactams
deoxygenation
Derivatives
preparation
fluorination
6 Citations (Scopus)

Asymmetric synthesis of chloroisothreonine derivatives via syn-stereoselective Mannich-type additions across N-sulfinyl-α- chloroimines

Callebaut, G., Colpaert, F., Nonn, M., Kiss, L., Sillanpää, R., Törnroos, K. W., Fülöp, F., De Kimpe, N. & Mangelinckx, S., jún. 7 2014, In : Organic and Biomolecular Chemistry. 12, 21, p. 3393-3405 13 p.

Research output: Article

esters
Esters
Derivatives
synthesis
Oxazolidinones
16 Citations (Scopus)

Compounds Blocking Methylglyoxal-induced Protein Modification and Brain Endothelial Injury

Tóth, A. E., Tóth, A., Walter, F. R., Kiss, L., Veszelka, S., Ózsvári, B., Puskás, L., Heimesaat, M. M., Dohgu, S., Kataoka, Y., Rákhely, G. & Deli, M., nov. 1 2014, In : Archives of Medical Research. 45, 8, p. 753-764 12 p.

Research output: Article

Pyruvaldehyde
Brain Injuries
Tretinoin
Proteins
Endothelial Cells
13 Citations (Scopus)
Esters
Phosphoranes
Derivatives
Amino Acids
Lactams
21 Citations (Scopus)

Sucrose esters increase drug penetration, but do not inhibit P-glycoprotein in Caco-2 intestinal epithelial cells

Kiss, L., Hellinger, É., Pilbat, A. M., Kittel, A., Tö Rök, Z., Furedi, Szakács, G., Veszelka, S., Sípos, P., Ózsvári, B. É., Puskás, L., Vastag, M., Szabó-Révész, P. & Deli, M., okt. 12 2014, In : Journal of Pharmaceutical Sciences. 103, 10, p. 3107-3119 13 p.

Research output: Article

P-Glycoprotein
Sucrose
Esters
Epithelial Cells
Pharmaceutical Preparations
121 Citations (Scopus)

Synthesis of carbocyclic and heterocyclic β-aminocarboxylic acids

Kiss, L. & Fülöp, F., jan. 22 2014, In : Chemical Reviews. 114, 2, p. 1116-1169 54 p.

Research output: Article

Heterocyclic Acids
Cyclic Amino Acids
Amino Acids
Derivatives
Amination
9 Citations (Scopus)
Lactams
Nucleophiles
Hydrides
Derivatives
Substrates
2013
37 Citations (Scopus)
High temperature reactors
Copper powder
Alkynes
Azides
Cycloaddition
24 Citations (Scopus)
Lactams
Amino acids
Derivatives
Amino Acids
2-norbornene
26 Citations (Scopus)
Triazoles
Derivatives
Acids
Copper powder
Azides
11 Citations (Scopus)

Efficient regio- and stereoselective access to novel fluorinated β-aminocyclohexanecarboxylates

Kiss, L., Nonn, M., Sillanpää, R., Fustero, S. & Fülöp, F., jún. 17 2013, In : Beilstein Journal of Organic Chemistry. 9, p. 1164-1169 6 p.

Research output: Article

Fluorine
Hydroxylation
Derivatives
Acids