Utilization of Copper-Catalyzed Carboarylation-Ring Closure for the Synthesis of New Oxazoline Derivatives

Ádám Sinai, Dóra Vangel, Tamás Gáti, P. Bombicz, Z. Novák

Research output: Contribution to journalArticle

25 Citations (Scopus)

Abstract

A copper-catalyzed carboarylation-ring-closure strategy was used for the modular synthesis of oxazolines via the reaction of 1-aryl- and 1-alkylpropargylamides and diaryliodonium salts. The novel approach enables the efficient, modular synthesis of oxazoline derivatives bearing fully substituted exo double bonds.

Original languageEnglish
Pages (from-to)4136-4139
Number of pages4
JournalOrganic Letters
Volume17
Issue number17
DOIs
Publication statusPublished - Aug 18 2015

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closures
Copper
Bearings (structural)
Salts
Derivatives
copper
rings
synthesis
salts

ASJC Scopus subject areas

  • Organic Chemistry
  • Physical and Theoretical Chemistry
  • Biochemistry

Cite this

Utilization of Copper-Catalyzed Carboarylation-Ring Closure for the Synthesis of New Oxazoline Derivatives. / Sinai, Ádám; Vangel, Dóra; Gáti, Tamás; Bombicz, P.; Novák, Z.

In: Organic Letters, Vol. 17, No. 17, 18.08.2015, p. 4136-4139.

Research output: Contribution to journalArticle

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