Synthesis of new 3-substituted aporphines

S. Berényi, C. Csutorás, S. Gyulai, G. Rusznyák

Research output: Contribution to journalArticle

6 Citations (Scopus)

Abstract

The methanesulfonic acid-induced rearrangement of 7-chloro-6-demethoxythebaine (10) in the presence of water or alcohols resulted in new 3-hydroxy-, or 3-alkoxy-11-hydroxy-10-methoxyaporphines (13, 14, 15, 16). O-Demethylation of the 3-methoxy derivative 14 with the methanesulfonic acid/methionine reagent-combination furnished 3,10,11-trihydroxyaporphine (18).

Original languageEnglish
Pages (from-to)1987-1992
Number of pages6
JournalSynthetic Communications
Volume31
Issue number13
DOIs
Publication statusPublished - 2001

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Aporphines
Methionine
Alcohols
Derivatives
Water
methanesulfonic acid

ASJC Scopus subject areas

  • Organic Chemistry

Cite this

Synthesis of new 3-substituted aporphines. / Berényi, S.; Csutorás, C.; Gyulai, S.; Rusznyák, G.

In: Synthetic Communications, Vol. 31, No. 13, 2001, p. 1987-1992.

Research output: Contribution to journalArticle

Berényi, S, Csutorás, C, Gyulai, S & Rusznyák, G 2001, 'Synthesis of new 3-substituted aporphines', Synthetic Communications, vol. 31, no. 13, pp. 1987-1992. https://doi.org/10.1081/SCC-100104415
Berényi, S. ; Csutorás, C. ; Gyulai, S. ; Rusznyák, G. / Synthesis of new 3-substituted aporphines. In: Synthetic Communications. 2001 ; Vol. 31, No. 13. pp. 1987-1992.
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