Synthesis of 6,7-Dibromoflavone and Its Regioselective Diversification via Suzuki–Miyaura Reactions

Sándor Jordán, Dávid Pajtás, T. Patonay, Peter Langer, Krisztina Kónya

Research output: Contribution to journalArticle

4 Citations (Scopus)

Abstract

The first synthesis pathway to 6,7-dibromoflavone and its transformations to 7-aryl-6-bromo- and 6,7-diarylflavones by Suzuki–Miyaura reactions are presented. Due to the different electronic effects of bromo substituents, the first attack proceeded with good site selectivity at position 7.

Original languageEnglish
JournalSynthesis (Germany)
DOIs
Publication statusAccepted/In press - Nov 20 2016

Keywords

  • catalysis
  • flavones
  • palladium
  • regioselectivity
  • Suzuki–Miyaura reaction

ASJC Scopus subject areas

  • Catalysis
  • Organic Chemistry

Cite this

Synthesis of 6,7-Dibromoflavone and Its Regioselective Diversification via Suzuki–Miyaura Reactions. / Jordán, Sándor; Pajtás, Dávid; Patonay, T.; Langer, Peter; Kónya, Krisztina.

In: Synthesis (Germany), 20.11.2016.

Research output: Contribution to journalArticle

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AU - Langer, Peter

AU - Kónya, Krisztina

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