Synthesis and reactions of paramagnetic aromatic aldehydes as useful synthetic building blocks

Research output: Contribution to journalArticle

1 Citation (Scopus)

Abstract

Starting from paramagnetic benzaldehyde, a benzophenone-type photoactivable spin label, paramagnetic warfarin and phenindione were synthesized. Nitration of protected benzylic alcohol led to 2-nitrobenzylmethanethiosulfonate, a thiol specific spin label, and 2-nitroaldehyde, which was a key compound for paramagnetic indigo, salicylic acid and nifedipine.

Original languageEnglish
Pages (from-to)2115-2120
Number of pages6
JournalSynthesis
Issue number13
DOIs
Publication statusPublished - Sep 6 2004

Fingerprint

Spin Labels
Aldehydes
Labels
Phenindione
Indigo Carmine
Nitration
Salicylic acid
Salicylic Acid
Warfarin
Nifedipine
Sulfhydryl Compounds
Alcohols
benzophenone
benzaldehyde

Keywords

  • Anticoagulant
  • Drugs
  • Free radicals
  • Indole
  • Pyridines

ASJC Scopus subject areas

  • Organic Chemistry

Cite this

Synthesis and reactions of paramagnetic aromatic aldehydes as useful synthetic building blocks. / Kálai, Tamás; Kulcsár, Gyozo; Jeko, József; Osz, Erzsébet; Hideg, Kálmán.

In: Synthesis, No. 13, 06.09.2004, p. 2115-2120.

Research output: Contribution to journalArticle

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