Synthesis and antibacterial activity of N-amino-derivatives of condensed pyridines

E. G. Paronikyan, Sh F. Hakobyan, A. S. Noravyan, G. Hajós, Sh Dashyan, R. V. Paronikyan, G. M. Stepanyan

Research output: Contribution to journalArticle

2 Citations (Scopus)

Abstract

A method based on condensed 4-cyanopyridinethiones using O-tosylhydroxylamine as the aminating agent was developed for preparing tosylates of N-amino-derivatives of pyrano[3,4-c]pyridines; 5,6,7,8- tetrahydroisoquinolines; and cyclopenta[c]pyridines. The antibacterial activity of the synthesized compounds was assessed.

Original languageEnglish
Pages (from-to)257-260
Number of pages4
JournalPharmaceutical Chemistry Journal
Volume47
Issue number5
DOIs
Publication statusPublished - Aug 2013

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Pyridines
Tetrahydroisoquinolines

Keywords

  • 5,6,7,8- tetrahydroisoquinolines
  • antibacterial activity
  • cyclopenta[c]pyridines
  • N-aminopyridines
  • pyrano[3,4-c]pyridines
  • tosylates

ASJC Scopus subject areas

  • Drug Discovery
  • Pharmacology

Cite this

Paronikyan, E. G., Hakobyan, S. F., Noravyan, A. S., Hajós, G., Dashyan, S., Paronikyan, R. V., & Stepanyan, G. M. (2013). Synthesis and antibacterial activity of N-amino-derivatives of condensed pyridines. Pharmaceutical Chemistry Journal, 47(5), 257-260. https://doi.org/10.1007/s11094-013-0940-3

Synthesis and antibacterial activity of N-amino-derivatives of condensed pyridines. / Paronikyan, E. G.; Hakobyan, Sh F.; Noravyan, A. S.; Hajós, G.; Dashyan, Sh; Paronikyan, R. V.; Stepanyan, G. M.

In: Pharmaceutical Chemistry Journal, Vol. 47, No. 5, 08.2013, p. 257-260.

Research output: Contribution to journalArticle

Paronikyan, EG, Hakobyan, SF, Noravyan, AS, Hajós, G, Dashyan, S, Paronikyan, RV & Stepanyan, GM 2013, 'Synthesis and antibacterial activity of N-amino-derivatives of condensed pyridines', Pharmaceutical Chemistry Journal, vol. 47, no. 5, pp. 257-260. https://doi.org/10.1007/s11094-013-0940-3
Paronikyan, E. G. ; Hakobyan, Sh F. ; Noravyan, A. S. ; Hajós, G. ; Dashyan, Sh ; Paronikyan, R. V. ; Stepanyan, G. M. / Synthesis and antibacterial activity of N-amino-derivatives of condensed pyridines. In: Pharmaceutical Chemistry Journal. 2013 ; Vol. 47, No. 5. pp. 257-260.
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