Simple and Condensed β-Lactams. Part 28. 1 the Synthesis of C-Methylcarumonams and of a Related Bis(carbamate)

J. Fetter, Ferenc Bertha, M. Kajtár-Peredy, Károly Lempert, Attila Sápi

Research output: Contribution to journalArticle

7 Citations (Scopus)

Abstract

Racemic carumonam analogues 2a-d are synthesised and found to be devoid of any bacterial activity; NaBH4 reduction of 18 affords both epimers of 8c with the (3RS,4RS)-4-[(1RS)] epirner as the main product, and cyclocondensation of phthalimidoacetyl chloride with racemic imine 14 gives rise to the formation of (3RS,4RS)-4-[(1RS)]-15 as a single epimer.

Original languageEnglish
Pages (from-to)118-119
Number of pages2
JournalJournal of Chemical Research - Part S
Issue number4
Publication statusPublished - 1997

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Lactams
Imines
Carbamates
Chlorides
carumonam

ASJC Scopus subject areas

  • Chemistry(all)

Cite this

Simple and Condensed β-Lactams. Part 28. 1 the Synthesis of C-Methylcarumonams and of a Related Bis(carbamate). / Fetter, J.; Bertha, Ferenc; Kajtár-Peredy, M.; Lempert, Károly; Sápi, Attila.

In: Journal of Chemical Research - Part S, No. 4, 1997, p. 118-119.

Research output: Contribution to journalArticle

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AU - Lempert, Károly

AU - Sápi, Attila

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