A one-pot process for palladium catalyzed direct C-H acylation of anilines in water using a removable ortho directing group

Fruzsina Szabó, Dániel Simkó, Z. Novák

Research output: Contribution to journalArticle

20 Citations (Scopus)

Abstract

A new mild, practical method for the synthesis of aminobenzophenone derivatives through a three step one-pot reaction sequence involving acylation of anilines, palladium catalyzed cross-dehydrogenative coupling of the formed anilides and the hydrolytic cleavage is reported. The full reaction sequence was performed under aqueous conditions.

Original languageEnglish
Pages (from-to)3883-3886
Number of pages4
JournalRSC Advances
Volume4
Issue number8
DOIs
Publication statusPublished - 2014

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Aniline Compounds
Anilides
Acylation
Palladium
Aniline
Derivatives
Hydrogen
Water

ASJC Scopus subject areas

  • Chemical Engineering(all)
  • Chemistry(all)

Cite this

A one-pot process for palladium catalyzed direct C-H acylation of anilines in water using a removable ortho directing group. / Szabó, Fruzsina; Simkó, Dániel; Novák, Z.

In: RSC Advances, Vol. 4, No. 8, 2014, p. 3883-3886.

Research output: Contribution to journalArticle

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